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Community harm-reduction information. Not medical advice. Content is available under the CC BY-SA 4.0 license.

GABA-A receptor positive allosteric modulator

34 substances share this mechanism of action.

GABA-A receptor positive allosteric modulator (General (no qualifier))1 GABA-A receptor positive allosteric modulator (barbiturate site)5 GABA-A receptor positive allosteric modulator (benzodiazepine site)25 GABA-A receptor positive allosteric modulator (binds to proconvulsant site)1 GABA-A receptor positive allosteric modulator (non-benzodiazepine site)1 GABA-A receptor positive allosteric modulator (preferential affinity for alpha-1, alpha-3, and alpha-5 subunits)1

GABA-A receptor positive allosteric modulator (general)

1 substance

GABAergic(1)

Carbamates(1)

Carisoprodol

GABA-A receptor positive allosteric modulator (barbiturate site)

5 substances

GABAergic(5)

Barbiturates(5)

Amobarbital
Pentobarbital
Phenobarbital
Secobarbital
Thiopental

GABA-A receptor positive allosteric modulator (benzodiazepine site)

25 substances

A-typical Hallucinogen(2)

Zolpidem
Zopiclone

GABAergic(23)

Common(5)

Alprazolam
Diazepam
Lorazepam
Oxazepam
Temazepam

Benzodiazepines(17)

Bromazepam
Brotizolam
Clonazepam
Delorazepam
Deschloroetizolam
Desmethylflunitrazepam
Diclazepam
Etizolam
Flualprazolam
Flubromazepam
Flubromazolam
Fluclotizolam
Flunitrazepam
Flunitrazolam
Midazolam
Pyrazolam
Triazolam

Thienodiazepine(1)

Metizolam

GABA-A receptor positive allosteric modulator (binds to proconvulsant site)

1 substance

Miscellaneous(1)

2M2B

GABA-A receptor positive allosteric modulator (non-benzodiazepine site)

1 substance

GABAergic(1)

Other GABAergics(1)

Kava

GABA-A receptor positive allosteric modulator (preferential affinity for alpha-1, alpha-3, and alpha-5 subunits)

1 substance

Miscellaneous(1)

Eszopiclone