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MK-801
Dizocilpine
Psychoactive Class
Dissociative
Hallucinogen
Chemical Class
Diarycycloheptene
Arylcyclohexyl-related NMDA antagonist
Contents
Dosage & Duration
Pharmacology
Harm Potential
Sources
Dosage & Duration
Oral
Dosage
Moderate
50-100 µg
Duration
After Effects
1-72 hours
Total
20-36 hours
Reagent Testing
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Pharmacology
Pharmacodynamics
Sources
Bluelight: MK-801 (4 mg sublingual) trip report
https://www.bluelight.org/community/threads/mk-801-4mg-sublingual-inexperienced-alice-in-wonderland-aint-got-nothin-on-this.846856/
Bluelight: MK-801 2.5 mg total (IM + rectal) trip report
https://www.bluelight.org/community/threads/mk-801-or-dizocilpine-dissociative.747376/
Erowid Experience: 3mg oral trip report
https://erowid.org/experiences/exp.php?ID=10737
Erowid Experience: IM dosing series
https://erowid.org/experiences/exp.php?ID=55729
Erowid Experience: The Most Beautiful Lobotomy I Ever Had
https://www.erowid.org/experiences/exp.php?ID=94476
TripSit: MK-801 Factsheet
https://tripbot.tripsit.me/factsheet/MK-801
Wikipedia
https://en.wikipedia.org/wiki/Dizocilpine
Wikipedia: Olney's lesions
https://en.wikipedia.org/wiki/Olney%27s_lesions
Further Reading
Clinical physiology and mechanism of dizocilpine (PMC)
https://pmc.ncbi.nlm.nih.gov/articles/PMC2835885/
Multiple-drug fatality case (MK-801 + benzodiazepines + alcohol)
https://pubmed.ncbi.nlm.nih.gov/12742697/
Plasma and brain half-life in rats (PubMed)
https://pubmed.ncbi.nlm.nih.gov/2540317/
11 sources cited